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- W4306154307 endingPage "2180" @default.
- W4306154307 startingPage "2180" @default.
- W4306154307 abstract "Erythromycin (ERY) is a macrolide compound with a broad antimicrobial spectrum which is currently being used to treat a large number of bacterial infections affecting the skin, respiratory tract, intestines, bones and other systems, proving great value from a clinical point of view. It became popular immediately after its discovery in 1952, due to its therapeutic effect against pathogens resistant to other drugs. Despite this major advantage, ERY exhibits several drawbacks, raising serious clinical challenges. Among them, the very low solubility in water and instability under acidic conditions cause a limited efficacy and bioavailability. Apart from this, higher doses promote drug resistance and undesirable effects. In order to overcome these disadvantages, during the past decades, a large variety of ERY formulations, including nanoparticles, have emerged. Despite the interest in ERY-(nano)formulations, a review on them is lacking. Therefore, this work was aimed at reviewing all efforts made to encapsulate ERY in formulations of various chemical compositions, sizes and morphologies. In addition, their preparation/synthesis, physico-chemical properties and performances were carefully analysed. Limitations of these studies, particularly the quantification of ERY, are discussed as well." @default.
- W4306154307 created "2022-10-14" @default.
- W4306154307 creator A5000743246 @default.
- W4306154307 creator A5007953899 @default.
- W4306154307 creator A5089698398 @default.
- W4306154307 date "2022-10-13" @default.
- W4306154307 modified "2023-10-18" @default.
- W4306154307 title "Erythromycin Formulations—A Journey to Advanced Drug Delivery" @default.
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