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- W4309089724 endingPage "7472" @default.
- W4309089724 startingPage "7472" @default.
- W4309089724 abstract "Antimicrobial resistance is a major public health issue raising growing concern in the face of dwindling response options. It is therefore urgent to find new anti-infective molecules enabling us to fight effectively against ever more numerous bacterial infections caused by ever more antibiotic-resistant bacteria. In this quest for new antibacterials, essential oils (or compounds extracted from essential oils) appear to be a promising therapeutic option. In the present work, we investigate the potential antibacterial synergy between a combination of terpinen-4-ol and α-terpineol (10:1) compared to standard tea tree oil. The minimum inhibitory concentration (MIC) and the minimum bactericidal concentration (MBC) were determined. Then, time kill assays, in vitro cytotoxicity and bactericidal activity on latent bacteria (persisters) were investigated. Finally, an in silico study of the pharmacokinetic parameters of α-terpineol was also performed. Altogether, our data demonstrate that the combination of terpinen-4-ol and α-terpineol might be a precious weapon to address ESKAPE pathogens." @default.
- W4309089724 created "2022-11-21" @default.
- W4309089724 creator A5051552050 @default.
- W4309089724 creator A5055132210 @default.
- W4309089724 creator A5074688010 @default.
- W4309089724 date "2022-11-02" @default.
- W4309089724 modified "2023-10-06" @default.
- W4309089724 title "First Evidence of a Combination of Terpinen-4-ol and α-Terpineol as a Promising Tool against ESKAPE Pathogens" @default.
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- W4309089724 doi "https://doi.org/10.3390/molecules27217472" @default.
- W4309089724 hasPubMedId "https://pubmed.ncbi.nlm.nih.gov/36364298" @default.
- W4309089724 hasPublicationYear "2022" @default.
- W4309089724 type Work @default.