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- W4310080087 abstract "Abstract This review describes the basic principles of radiometal-theranostics and its dawn based on the development of the positron-emitting 86 Y and 86 Y-labeled radiopharmaceuticals to quantify biodistribution and dosimetry of 90 Y-labeled analogue therapeutics. The nuclear and inorganic development of 86 Y (including nuclear and cross section data, irradiation, radiochemical separation and recovery) led to preclinical and clinical evaluation of 86 Y-labeled citrate and EDTMP complexes and yielded organ radiation doses in terms of mGy/MBq 90 Y. The approach was extended to [ 86/90 Y]Y-DOTA-TOC, yielding again yielded organ radiation doses in terms of mGy/MBq 90 Y. The review further discusses the consequences of this early development in terms of further radiometals that were used ( 68 Ga, 177 Lu etc.), more chelators that were developed, new biological targets that were addressed (SSTR, PSMA, FAP, etc.) and subsequent generations of radiometal-theranostics that resulted out of that." @default.
- W4310080087 created "2022-11-30" @default.
- W4310080087 creator A5037619007 @default.
- W4310080087 creator A5064057435 @default.
- W4310080087 date "2022-11-24" @default.
- W4310080087 modified "2023-09-30" @default.
- W4310080087 title "Radiometal-theranostics: the first 20 years*" @default.
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