Matches in SemOpenAlex for { <https://semopenalex.org/work/W4313251237> ?p ?o ?g. }
- W4313251237 endingPage "e236" @default.
- W4313251237 startingPage "e223" @default.
- W4313251237 abstract "Anaplastic lymphoma kinase (ALK) is one of the most popular targets for anticancer therapies. In the past decade, the use of anaplastic lymphoma tyrosine kinase inhibitors (ALK-TKIs), including crizotinib and ceritinib, has been a reliable and standard options for patients with lung cancer, particularly for patients with nonsmall cell lung carcinoma. ALK-targeted therapies initially benefit the patients, yet, resistance eventually occurs. Therefore, resistance mechanisms of ALK-TKIs and the solutions have become a formidable challenge in the development of ALK inhibitors. In this review, based on the knowledge of reported ALK inhibitors, we illustrated the crystal structures of ALK, summarized the resistance mechanisms of ALK-targeted drugs, and proposed potential therapeutic strategies to prevent or overcome the resistance." @default.
- W4313251237 created "2023-01-06" @default.
- W4313251237 creator A5004693417 @default.
- W4313251237 creator A5006816564 @default.
- W4313251237 creator A5032426102 @default.
- W4313251237 creator A5045839676 @default.
- W4313251237 creator A5067614579 @default.
- W4313251237 creator A5068850994 @default.
- W4313251237 date "2022-12-01" @default.
- W4313251237 modified "2023-09-26" @default.
- W4313251237 title "Hallmarks of Anaplastic Lymphoma Kinase Inhibitors with Its Quick Emergence of Drug Resistance" @default.
- W4313251237 cites W1489468742 @default.
- W4313251237 cites W1519176158 @default.
- W4313251237 cites W1528343569 @default.
- W4313251237 cites W1963822859 @default.
- W4313251237 cites W1964924351 @default.
- W4313251237 cites W1966319894 @default.
- W4313251237 cites W1969391810 @default.
- W4313251237 cites W1981872831 @default.
- W4313251237 cites W1995274368 @default.
- W4313251237 cites W1995641421 @default.
- W4313251237 cites W1997476230 @default.
- W4313251237 cites W2001171502 @default.
- W4313251237 cites W2005841386 @default.
- W4313251237 cites W2008167816 @default.
- W4313251237 cites W2008570836 @default.
- W4313251237 cites W2010978319 @default.
- W4313251237 cites W2014795318 @default.
- W4313251237 cites W2018336040 @default.
- W4313251237 cites W2018416379 @default.
- W4313251237 cites W2021876472 @default.
- W4313251237 cites W2022354436 @default.
- W4313251237 cites W2023513814 @default.
- W4313251237 cites W2026247210 @default.
- W4313251237 cites W2027337735 @default.
- W4313251237 cites W2031714712 @default.
- W4313251237 cites W2035282066 @default.
- W4313251237 cites W2038053082 @default.
- W4313251237 cites W2038586807 @default.
- W4313251237 cites W2038665105 @default.
- W4313251237 cites W2041490232 @default.
- W4313251237 cites W2041723408 @default.
- W4313251237 cites W2044558623 @default.
- W4313251237 cites W2052016211 @default.
- W4313251237 cites W2054445623 @default.
- W4313251237 cites W2055402151 @default.
- W4313251237 cites W2056148235 @default.
- W4313251237 cites W2059122821 @default.
- W4313251237 cites W2060275730 @default.
- W4313251237 cites W2066266086 @default.
- W4313251237 cites W2071089074 @default.
- W4313251237 cites W2075280221 @default.
- W4313251237 cites W2080992857 @default.
- W4313251237 cites W2082020673 @default.
- W4313251237 cites W2096156234 @default.
- W4313251237 cites W2097417052 @default.
- W4313251237 cites W2106915761 @default.
- W4313251237 cites W2109770623 @default.
- W4313251237 cites W2113327188 @default.
- W4313251237 cites W2113800457 @default.
- W4313251237 cites W2114256922 @default.
- W4313251237 cites W2117809853 @default.
- W4313251237 cites W2123394258 @default.
- W4313251237 cites W2123727052 @default.
- W4313251237 cites W2126298634 @default.
- W4313251237 cites W2140333474 @default.
- W4313251237 cites W2145165647 @default.
- W4313251237 cites W2146396128 @default.
- W4313251237 cites W2153782264 @default.
- W4313251237 cites W2155405367 @default.
- W4313251237 cites W2168691181 @default.
- W4313251237 cites W2170144893 @default.
- W4313251237 cites W2473726601 @default.
- W4313251237 cites W2530539219 @default.
- W4313251237 cites W2548979713 @default.
- W4313251237 cites W2553908226 @default.
- W4313251237 cites W2607398004 @default.
- W4313251237 cites W2616239758 @default.
- W4313251237 cites W2765258454 @default.
- W4313251237 cites W2766746980 @default.
- W4313251237 cites W2788006464 @default.
- W4313251237 cites W2794623623 @default.
- W4313251237 cites W2883124357 @default.
- W4313251237 cites W2884617673 @default.
- W4313251237 cites W2908885437 @default.
- W4313251237 cites W2942185172 @default.
- W4313251237 cites W2954565338 @default.
- W4313251237 cites W2969431490 @default.
- W4313251237 cites W2969467314 @default.
- W4313251237 cites W2971320546 @default.
- W4313251237 cites W2978074062 @default.
- W4313251237 cites W2990222327 @default.
- W4313251237 cites W2996380129 @default.
- W4313251237 cites W2997993855 @default.
- W4313251237 cites W3007665819 @default.
- W4313251237 cites W3008159666 @default.
- W4313251237 cites W3055236141 @default.
- W4313251237 cites W3083635816 @default.