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- W4313531431 endingPage "115052" @default.
- W4313531431 startingPage "115052" @default.
- W4313531431 abstract "The purinergic signaling has drawn attention from academia and more recently from pharmaceutical industries as a potential therapeutic route for cancer treatment, since ATP may act as chemotactic agent and possess in vitro antineoplastic activity. On the other way, adenosine, produced in extracellular medium by ecto-5'-NT, acts as immunosuppressor and is related to neoangiogenesis, vasculogenesis and evasion to the immune system. Consequently, inhibitors of ecto-5'-NT may prevent tumor progression, reducing adenosine concentrations, preventing escape from the host's immune system and slowing cancer's growth. This review aims to highlight important biochemical and structural features of ecto-5'NT, highlight its expression profile in normal and cancer cell lines detailing compounds which may act as expression regulators and to review the several classes of ecto-5'NT inhibitors developed in the past 12 years, in order to build a general structure-activity relationship model to guide further compound design." @default.
- W4313531431 created "2023-01-06" @default.
- W4313531431 creator A5016260523 @default.
- W4313531431 creator A5018978631 @default.
- W4313531431 creator A5049562552 @default.
- W4313531431 creator A5062748725 @default.
- W4313531431 creator A5079325248 @default.
- W4313531431 date "2023-02-01" @default.
- W4313531431 modified "2023-10-18" @default.
- W4313531431 title "Targeting ecto-5′-nucleotidase: A comprehensive review into small molecule inhibitors and expression modulators" @default.
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