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- W4362457925 startingPage "146" @default.
- W4362457925 abstract "Bortezomib (BTZ) is a first-in-class reversible and selective proteasome inhibitor. It inhibits the ubiquitin proteasome pathway that leads to the degradation of many intracellular proteins. Initially, BTZ was FDA approved for the treatment of refractory or relapsed multiple myeloma (MM) in 2003. Later, its usage was approved for patients with previously untreated MM. In 2006, BTZ was approved for the treatment of relapsed or refractory Mantle Cell Lymphoma (MCL) and, in 2014, for previously untreated MCL. BTZ has been extensively studied either alone or in combination with other drugs for the treatment of different liquid tumors especially in MM. However, limited data evaluated the efficacy and safety of using BTZ in patients with solid tumors. In this review, we will discuss the advanced and novel mechanisms of action of BTZ documented in MM, solid tumors and liquid tumors. Moreover, we will shed the light on the newly discovered pharmacological effects of BTZ in other prevalent diseases." @default.
- W4362457925 created "2023-04-05" @default.
- W4362457925 creator A5005814577 @default.
- W4362457925 creator A5011094456 @default.
- W4362457925 creator A5064060272 @default.
- W4362457925 creator A5068569741 @default.
- W4362457925 creator A5074450777 @default.
- W4362457925 date "2023-01-01" @default.
- W4362457925 modified "2023-09-26" @default.
- W4362457925 title "Bortezomib advanced mechanisms of action in multiple myeloma, solid and liquid tumors along with its novel therapeutic applications." @default.
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