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- W4362621697 abstract "<p>PDF file - 1250K, Supplementary Figure S1: SC144 exhibits cytotoxicity in human ovarian cancer cell lines; Supplementary Figure S2: Confirmation of gp130 protein expression, glycosylation phosphorylation and internalization; Supplementary Figure S3: Constitutive Stat3 (Tyr705) phosphorylation is gp130 dependent; Supplementary Figure S4: gp130/Stat3 knockdown suppresses the expression of downstream genes; Supplementary Figure S5: SC144's effects on pancreatic cancer cells; Supplementary Figure S6: Gp130/Stat3 inhibition causes cytotoxicity in ovarian cancer cells; Supplementary Figure S7: SC144 inhibits cytokine-induced Stat3 activation; Supplementary Figure S8: SC144 treatment did not cause systemic toxicity.</p>" @default.
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- W4362621697 date "2023-04-03" @default.
- W4362621697 modified "2023-09-27" @default.
- W4362621697 title "Supplementary Figures 1 - 8 from Discovery of a Novel Orally Active Small-Molecule gp130 Inhibitor for the Treatment of Ovarian Cancer" @default.
- W4362621697 doi "https://doi.org/10.1158/1535-7163.22501387.v1" @default.
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