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- W4365457915 endingPage "108414" @default.
- W4365457915 startingPage "108414" @default.
- W4365457915 abstract "Lysophosphatidic acid (LPA) is a bioactive lipid mediator that regulates a variety of cellular functions such as cell proliferation, migration, survival, calcium mobilization, cytoskeletal rearrangements, and neurite retraction. The biological actions of LPA are mediated by at least six G protein-coupled receptors known as LPAR1-6. Given that LPAR1-3 were among the first LPARs identified, the majority of research efforts have focused on understanding their biology. This review provides an in-depth discussion of LPAR5, which has recently emerged as a key player in regulating normal intestinal homeostasis and modulating pathological conditions such as pain, itch, inflammatory diseases, and cancer. We also present a chronological overview of the efforts made to develop compounds that target LPAR5 for use as tool compounds to probe or validate LPAR5 biology and therapeutic agents for the treatment of inflammatory diseases and cancer." @default.
- W4365457915 created "2023-04-15" @default.
- W4365457915 creator A5032960258 @default.
- W4365457915 creator A5057108769 @default.
- W4365457915 creator A5071553204 @default.
- W4365457915 creator A5077058937 @default.
- W4365457915 date "2023-05-01" @default.
- W4365457915 modified "2023-10-16" @default.
- W4365457915 title "Emerging roles of lysophosphatidic acid receptor subtype 5 (LPAR5) in inflammatory diseases and cancer" @default.
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