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- W4378550010 abstract "The protein that forms the inner shell of the HBV virus, known as the capsid core protein, plays a crucial role in allowing chronic HBV infections to persist. Studies have shown that disrupting the assembly of the capsid can effectively combat the virus, and small molecule drugs that target the HBV capsid assembly modulator (CAM) process have been successful in clinical trials. Herein is described a distinct series of di-fluoro azepane CAMs with exceptional potency, pharmacokinetic, and solubility properties." @default.
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- W4378550010 date "2023-08-01" @default.
- W4378550010 modified "2023-10-01" @default.
- W4378550010 title "Di-fluoro azepane HBV capsid assembly modulators" @default.
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- W4378550010 doi "https://doi.org/10.1016/j.bmcl.2023.129350" @default.
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