Matches in SemOpenAlex for { <https://semopenalex.org/work/W4378781929> ?p ?o ?g. }
- W4378781929 endingPage "334" @default.
- W4378781929 startingPage "326" @default.
- W4378781929 abstract "Antibiotic resistance (AR) is a silent pandemic that kills millions worldwide. Although the development of new therapeutic agents against antibiotic resistance is in urgent demand, this has presented a great challenge, especially for Gram-negative bacteria that have inherent drug-resistance mediated by impermeable outer membranes and multidrug efflux pumps that actively extrude various drugs from the bacteria. For the last two decades, multidrug efflux pumps, including AcrAB-TolC, the most clinically important efflux pump in Gram-negative bacteria, have drawn great attention as strategic targets for re-sensitizing bacteria to the existing antibiotics. This article aims to provide a concise overview of the AcrAB-TolC operational mechanism, reviewing its architecture and substrate specificity, as well as the recent development of AcrAB-TolC inhibitors. [BMB Reports 2023; 56(6): 326-334]." @default.
- W4378781929 created "2023-06-01" @default.
- W4378781929 creator A5027044660 @default.
- W4378781929 date "2023-06-07" @default.
- W4378781929 modified "2023-10-14" @default.
- W4378781929 title "AcrAB-TolC, a major efflux pump in Gram negative bacteria: toward understanding its operation mechanism" @default.
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