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- W4380992016 abstract "Peroxisome proliferative activated receptors (PPARs) act as ligand-activated transcription factors involved in glucose and lipoprotein metabolism, and in inflammation. binding to specific response elements (PPREs) within the nucleus. Heterodimerization with a retinoid X receptor and interaction with coactivators and corepressors occur after binding of natural or synthetic agonists. The first synthetic agonists in clinical use were fibrates for PPAR alpha and thiazolidinediones for PPAR gamma. Dual α γ agonists, pan α γ δ agonists, partial agonists or selective PPAR modulators (SPPARMs) have been evaluated in clinical development in diabetic people with current stage prior or after marketing authorization tabulated." @default.
- W4380992016 created "2023-06-17" @default.
- W4380992016 creator A5087106254 @default.
- W4380992016 date "2023-01-01" @default.
- W4380992016 modified "2023-09-23" @default.
- W4380992016 title "The PPAR System in Diabetes" @default.
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