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- W4382068648 endingPage "1815" @default.
- W4382068648 startingPage "1815" @default.
- W4382068648 abstract "The indole heterocycle represents one of the most important scaffolds in medicinal chemistry and is shared among a number of drugs clinically used in different therapeutic areas. Due to its varied biological activities, high unique chemical properties and significant pharmacological behaviors, indole derivatives have drawn considerable interest in the last decade as antitumor agents active against different types of cancers. The research of novel antiproliferative drugs endowed with enhanced efficacy and reduced toxicity led to the approval by U.S. Food and Drug Administration of the indole-based anticancer agents Sunitinib, Nintedanib, Osimertinib, Panobinostat, Alectinib and Anlotinib. Additionally, new drug delivery systems have been developed to protect the active principle from degradation and to direct the drug to the specific site for clinical use, thus reducing its toxicity. In the present work is an updated review of the recently approved indole-based anti-cancer agents and the nanotechnology systems developed for their delivery." @default.
- W4382068648 created "2023-06-27" @default.
- W4382068648 creator A5022877107 @default.
- W4382068648 creator A5048118855 @default.
- W4382068648 creator A5058428207 @default.
- W4382068648 creator A5081580744 @default.
- W4382068648 creator A5091202892 @default.
- W4382068648 creator A5092268553 @default.
- W4382068648 date "2023-06-25" @default.
- W4382068648 modified "2023-10-14" @default.
- W4382068648 title "Indole Antitumor Agents in Nanotechnology Formulations: An Overview" @default.
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