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- W4382559650 endingPage "115613" @default.
- W4382559650 startingPage "115613" @default.
- W4382559650 abstract "Many populations worldwide are suffering from central nervous system (CNS) diseases such as brain tumors, neurodegenerative diseases (Alzheimer's disease, Parkinson's disease and Huntington's disease) and stroke. There is a shortage of effective drugs for most CNS diseases. As one of the regulatory mechanisms of epigenetics, the particular role and therapeutic benefits of histone deacetylases (HDACs) in the CNS have been extensively studied. In recent years, HDACs have attracted increasing attention as potential drug targets for CNS diseases. In this review, we summarize the recent applications of representative histone deacetylases inhibitors (HDACis) in CNS diseases and discuss the challenges in developing HDACis with different structures and better blood-brain barrier (BBB) permeability, hoping to promote the development of more effective bioactive HDACis for the treatment of CNS diseases." @default.
- W4382559650 created "2023-06-30" @default.
- W4382559650 creator A5004724436 @default.
- W4382559650 creator A5040648061 @default.
- W4382559650 creator A5053467487 @default.
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- W4382559650 creator A5068986165 @default.
- W4382559650 creator A5080209274 @default.
- W4382559650 creator A5084282171 @default.
- W4382559650 date "2023-10-01" @default.
- W4382559650 modified "2023-09-26" @default.
- W4382559650 title "Perspectives and new aspects of histone deacetylase inhibitors in the therapy of CNS diseases" @default.
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