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- W4383375364 abstract "Azanucleosides, such as 5-azacytidine and decitabine, are DNA demethylating agents used in the treatment of acute myeloid leukemia and myelodysplastic syndromes. Researchers continue to explore their utility in the treatment of other hematologic and solid tumors. Based on the capacity of the compounds to inhibit DNA methyltransferase enzymes and the important role of DNA methylation in health and disease, it is essential to understand the molecular changes that azanucleosides induce and how these changes may improve treatment outcomes in subsets of patients. This review summarizes the molecular and therapeutic actions of azanucleosides and discusses recent clinical trials of these compounds as single agents or in combination therapy for the treatment of cancer and related conditions." @default.
- W4383375364 created "2023-07-07" @default.
- W4383375364 creator A5047899936 @default.
- W4383375364 creator A5092414671 @default.
- W4383375364 date "2023-07-05" @default.
- W4383375364 modified "2023-09-26" @default.
- W4383375364 title "Therapeutic Applications of Azanucleoside Analogs as DNA Demethylating Agents" @default.
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- W4383375364 doi "https://doi.org/10.3390/epigenomes7030012" @default.
- W4383375364 hasPubMedId "https://pubmed.ncbi.nlm.nih.gov/37489400" @default.
- W4383375364 hasPublicationYear "2023" @default.
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