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- W4384023963 endingPage "1119" @default.
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- W4384023963 abstract "Targets play an indispensable and pivotal role in the development of radiopharmaceuticals. However, the initial stages of drug discovery projects are often plagued by frequent failures due to inadequate information on druggability and suboptimal target selection. In this context, we aim to present a comprehensive review of the factors that influence target druggability for diagnostic radiopharmaceuticals. Specifically, we explore the crucial determinants of target specificity, abundance, localization, and positivity rate and their respective implications. Through a detailed analysis of existing protein targets, we elucidate the significance of each factor. By carefully considering and balancing these factors during the selection of targets, more efficacious and targeted radiopharmaceuticals are expected to be designed for the diagnosis of a wide range of diseases in the future." @default.
- W4384023963 created "2023-07-13" @default.
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- W4384023963 date "2023-07-12" @default.
- W4384023963 modified "2023-10-16" @default.
- W4384023963 title "Druggability of Targets for Diagnostic Radiopharmaceuticals" @default.
- W4384023963 cites W1490266165 @default.
- W4384023963 cites W1522571942 @default.
- W4384023963 cites W1606142774 @default.
- W4384023963 cites W1840512156 @default.
- W4384023963 cites W188996788 @default.
- W4384023963 cites W1923415348 @default.
- W4384023963 cites W1926568554 @default.
- W4384023963 cites W193225678 @default.
- W4384023963 cites W1968408292 @default.
- W4384023963 cites W1970225047 @default.
- W4384023963 cites W1973268693 @default.
- W4384023963 cites W1981502499 @default.
- W4384023963 cites W1983042517 @default.
- W4384023963 cites W1989215781 @default.
- W4384023963 cites W1995160345 @default.
- W4384023963 cites W1997890450 @default.
- W4384023963 cites W2001466921 @default.
- W4384023963 cites W2001858363 @default.
- W4384023963 cites W2003137271 @default.
- W4384023963 cites W2007843828 @default.
- W4384023963 cites W2012034410 @default.
- W4384023963 cites W2023096047 @default.
- W4384023963 cites W2024078329 @default.
- W4384023963 cites W2024882352 @default.
- W4384023963 cites W2034176597 @default.
- W4384023963 cites W2035278976 @default.
- W4384023963 cites W2040935952 @default.
- W4384023963 cites W2043680485 @default.
- W4384023963 cites W2048952941 @default.
- W4384023963 cites W2054912906 @default.
- W4384023963 cites W2060220993 @default.
- W4384023963 cites W2060244348 @default.
- W4384023963 cites W2060729557 @default.
- W4384023963 cites W2062949575 @default.
- W4384023963 cites W2063576864 @default.
- W4384023963 cites W2066735646 @default.
- W4384023963 cites W2067637906 @default.
- W4384023963 cites W2071384955 @default.
- W4384023963 cites W2072171721 @default.
- W4384023963 cites W2076570311 @default.
- W4384023963 cites W2077172876 @default.
- W4384023963 cites W2078620068 @default.
- W4384023963 cites W2084864412 @default.
- W4384023963 cites W2089275510 @default.
- W4384023963 cites W2094229819 @default.
- W4384023963 cites W2103126725 @default.
- W4384023963 cites W2107271788 @default.
- W4384023963 cites W2110601381 @default.
- W4384023963 cites W2114200547 @default.
- W4384023963 cites W2114634539 @default.
- W4384023963 cites W2116531960 @default.
- W4384023963 cites W2122767481 @default.
- W4384023963 cites W2127363066 @default.
- W4384023963 cites W2127896250 @default.
- W4384023963 cites W2131480828 @default.
- W4384023963 cites W2142892314 @default.
- W4384023963 cites W2145728390 @default.
- W4384023963 cites W2146384083 @default.
- W4384023963 cites W2155421560 @default.
- W4384023963 cites W2156921812 @default.
- W4384023963 cites W2158407564 @default.
- W4384023963 cites W2159821105 @default.
- W4384023963 cites W2165946747 @default.
- W4384023963 cites W2167064996 @default.
- W4384023963 cites W2171234688 @default.
- W4384023963 cites W2260663127 @default.
- W4384023963 cites W2287868019 @default.
- W4384023963 cites W2290598353 @default.
- W4384023963 cites W2315407377 @default.
- W4384023963 cites W2339631364 @default.
- W4384023963 cites W2339880566 @default.
- W4384023963 cites W2340761255 @default.
- W4384023963 cites W2519418984 @default.
- W4384023963 cites W2554140915 @default.
- W4384023963 cites W2560407658 @default.
- W4384023963 cites W2560808776 @default.
- W4384023963 cites W2594098019 @default.
- W4384023963 cites W2597816781 @default.
- W4384023963 cites W2604465368 @default.
- W4384023963 cites W2607721315 @default.
- W4384023963 cites W2611296537 @default.
- W4384023963 cites W2613629789 @default.
- W4384023963 cites W2621105275 @default.
- W4384023963 cites W2771996063 @default.
- W4384023963 cites W2772609666 @default.
- W4384023963 cites W2785428883 @default.