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- W4385587744 endingPage "146" @default.
- W4385587744 startingPage "117" @default.
- W4385587744 abstract "Oxazolidinone scaffolds have a significant role in drug discovery and development. Compounds with an oxazolidinone skeleton have a wide range of pharmacologic effects and are used to treat bacterial infection. The fully synthetic oxazolidinone antibacterial drugs linezolid and tedizolid have proven clinical therapeutic benefits with the emergence and evolution of resistant bacteria. Antibacterial drugs containing oxazolidinone have several advantages, including favorable pharmacokinetics and pharmacodynamics, novel antibacterial pathways, and druggability. Here, we focus on oxazolidinones derived from structural modifications of linezolid and other possible oxazolidinone drugs, describing their structure–activity relationships, druggability, and safety, and providing a unique idea for improving more potent and safer oxazolidinone drugs." @default.
- W4385587744 created "2023-08-05" @default.
- W4385587744 creator A5022315541 @default.
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- W4385587744 creator A5060296554 @default.
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- W4385587744 creator A5073501391 @default.
- W4385587744 date "2023-01-01" @default.
- W4385587744 modified "2023-09-24" @default.
- W4385587744 title "Oxazolidinone scaffolds in drug discovery and development" @default.
- W4385587744 cites W1552315958 @default.
- W4385587744 cites W1565970806 @default.
- W4385587744 cites W1859276716 @default.
- W4385587744 cites W1967767172 @default.
- W4385587744 cites W1969304488 @default.
- W4385587744 cites W1972821355 @default.
- W4385587744 cites W1980595924 @default.
- W4385587744 cites W1984051860 @default.
- W4385587744 cites W1985895918 @default.
- W4385587744 cites W1990362340 @default.
- W4385587744 cites W1990661343 @default.
- W4385587744 cites W1992157577 @default.
- W4385587744 cites W1998002492 @default.
- W4385587744 cites W1999979510 @default.
- W4385587744 cites W2001147671 @default.
- W4385587744 cites W2009662699 @default.
- W4385587744 cites W2017662055 @default.
- W4385587744 cites W2022937061 @default.
- W4385587744 cites W2027155313 @default.
- W4385587744 cites W2032955926 @default.
- W4385587744 cites W2039756687 @default.
- W4385587744 cites W2039989497 @default.
- W4385587744 cites W2043070998 @default.
- W4385587744 cites W2044768462 @default.
- W4385587744 cites W2047642255 @default.
- W4385587744 cites W2048747882 @default.
- W4385587744 cites W2051979560 @default.
- W4385587744 cites W2054762986 @default.
- W4385587744 cites W2055547621 @default.
- W4385587744 cites W2060839079 @default.
- W4385587744 cites W2067771624 @default.
- W4385587744 cites W2068051461 @default.
- W4385587744 cites W2068204518 @default.
- W4385587744 cites W2068398959 @default.
- W4385587744 cites W2071342482 @default.
- W4385587744 cites W2074503128 @default.
- W4385587744 cites W2082395198 @default.
- W4385587744 cites W2084341599 @default.
- W4385587744 cites W2089881428 @default.
- W4385587744 cites W2090816462 @default.
- W4385587744 cites W2092196558 @default.
- W4385587744 cites W2092973221 @default.
- W4385587744 cites W2098997185 @default.
- W4385587744 cites W2104671122 @default.
- W4385587744 cites W2106330783 @default.
- W4385587744 cites W2108106379 @default.
- W4385587744 cites W2109736604 @default.
- W4385587744 cites W2109824815 @default.
- W4385587744 cites W2111236190 @default.
- W4385587744 cites W2117892088 @default.
- W4385587744 cites W2119704253 @default.
- W4385587744 cites W2123162658 @default.
- W4385587744 cites W2124788857 @default.
- W4385587744 cites W2126221698 @default.
- W4385587744 cites W2128076923 @default.
- W4385587744 cites W2130282734 @default.
- W4385587744 cites W2143206150 @default.
- W4385587744 cites W2143949361 @default.
- W4385587744 cites W2143968171 @default.
- W4385587744 cites W2145514220 @default.
- W4385587744 cites W2145596140 @default.
- W4385587744 cites W2149375508 @default.
- W4385587744 cites W2151742889 @default.
- W4385587744 cites W2151859311 @default.
- W4385587744 cites W2155258790 @default.
- W4385587744 cites W2160434710 @default.
- W4385587744 cites W2163224809 @default.
- W4385587744 cites W2165473666 @default.
- W4385587744 cites W2167713581 @default.
- W4385587744 cites W2168281308 @default.
- W4385587744 cites W2168635615 @default.
- W4385587744 cites W2170367123 @default.
- W4385587744 cites W2171026842 @default.
- W4385587744 cites W2171998389 @default.
- W4385587744 cites W2179122606 @default.
- W4385587744 cites W2250661867 @default.
- W4385587744 cites W2276171955 @default.
- W4385587744 cites W2276443311 @default.
- W4385587744 cites W2312584567 @default.
- W4385587744 cites W2320285551 @default.
- W4385587744 cites W2321174248 @default.
- W4385587744 cites W2329336725 @default.
- W4385587744 cites W2330393631 @default.
- W4385587744 cites W2340901723 @default.
- W4385587744 cites W2405699446 @default.
- W4385587744 cites W2418293022 @default.