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- W49029705 abstract "OBJECTIVE Nicotinic acetylcholine receptors (nAChRs) are important for inhibition of inflammation. Agonists of the alpha-7 subunit demonstrate anti-inflammatory activity both in vitro and in vivo. The purpose of this study was to test the anti-inflammatory effect of CTI-78, a specific agonist of alpha-7 with an IC50=225nM, in a rodent model of acute inflammation. METHODS The rat carrageenan-induced paw edema model was used to evaluate the anti-inflammatory effects of alpha-7 agonists. CTI-78 was prophylactically dosed at 10, 4, or 1 mg/kg, intraperitoneally. Indomethacin, a clinically relevant nonsteroidal anti-inflammatory drug, was used as an internal reference control. RESULTS CTI-78 inhibited paw edema at a range of 9–31% at 10mg/kg over the course of the study (1–5 hours). CONCLUSION CTI-78, a specific alpha-7 agonist, inhibits paw inflammation induced by carrageenan." @default.
- W49029705 created "2016-06-24" @default.
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- W49029705 date "2006-03-01" @default.
- W49029705 modified "2023-09-27" @default.
- W49029705 title "Anti‐Inflammatory Effects of Alpha‐7 Nicotinic Cholinergic Receptor Agonists in Rat Carrageenan‐Induced Paw Edema" @default.
- W49029705 doi "https://doi.org/10.1096/fasebj.20.5.a1127-d" @default.
- W49029705 hasPublicationYear "2006" @default.
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