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- W53238597 abstract "Neuropeptides seem to play critical roles in the modulation of anxiety and in the pathophysiology of anxiety disorders. Specific, small-molecule, non-peptide receptor ligands targeting these peptide systems have been developed and are at various stages of the drug development process, such as antagonists acting at the corticotropin-releasing factor, cholecystokinin, neurokinin, neuropeptide Y, vasopressin, melanocortin, angiotensin, galanin, bombesin, or melanin-stimulating hormone receptors. Furthermore, oxytocin, δ-opiate, and orphanin FQ/nociceptin receptor agonists have been developed and shown to have anxiolytic-like properties in preclinical models. Some of these compounds are currently in clinical testing. This review provides an update of the preclinical and clinical status of the field. Although a number of obstacles need to be overcome in this area, it can be concluded that compounds acting at neuropeptide targets represents a highly promising approach for the development of the next generation drugs to treat anxiety disorders." @default.
- W53238597 created "2016-06-24" @default.
- W53238597 creator A5040568010 @default.
- W53238597 date "2008-01-01" @default.
- W53238597 modified "2023-09-25" @default.
- W53238597 title "Chapter 4.1 Peptide receptor ligands to treat anxiety disorders" @default.
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