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- W5845191 endingPage "320" @default.
- W5845191 startingPage "281" @default.
- W5845191 abstract "The Kelch-like ECH-associated protein 1 (Keap1)-nuclear factor E2-related factor 2 (Nrf2) pathway is one of the major signaling cascades involved in cell defense and survival against endogenous and exogenous stress. While Nrf2 and its target genes provide protection against various age-related diseases including tumorigenesis, constitutively active Nrf2 in cancer cells increases the expression of cytoprotective genes and, consequently, enhances proliferation via metabolic reprogramming and inhibition of apoptosis. Herein, we review the current understanding of the regulation of Nrf2 in normal cells as well as its dual role in cancer. Furthermore, the mechanisms of Nrf2 dysregulation in cancer, consequences of unchecked Nrf2 activity, and therapies targeting the Keap1-Nrf2 system are discussed." @default.
- W5845191 created "2016-06-24" @default.
- W5845191 creator A5001075589 @default.
- W5845191 creator A5031300613 @default.
- W5845191 creator A5074126248 @default.
- W5845191 creator A5080117485 @default.
- W5845191 creator A5090216995 @default.
- W5845191 date "2014-01-01" @default.
- W5845191 modified "2023-10-18" @default.
- W5845191 title "Role of the Keap1–Nrf2 Pathway in Cancer" @default.
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