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- W64035408 endingPage "223" @default.
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- W64035408 abstract "Abstract Fruits and vegetables are known to possess chemopreventive activities in the fight against cancer. Some active metabolites have been fully characterized and were found to have epigenetic bioactivities such as inhibition of DNA methylation. Among them, polyphenols have demonstrated potent DNA methyltransferase (DNMT) activity. This activity is associated with DNA demethylation at the CpG islands and the reactivation of silenced genes involved in the methylation process. We review here the relevant published literature focusing on natural polyphenols and their relationship with epigenetic modifications particularly on DNMT. Indeed, some of them like Epigallocatechin-3-gallate appear as a promising DNMT inhibitor, while the mode of action of other polyphenols remains to be deciphered." @default.
- W64035408 created "2016-06-24" @default.
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- W64035408 creator A5088767601 @default.
- W64035408 creator A5089211056 @default.
- W64035408 date "2014-01-01" @default.
- W64035408 modified "2023-09-26" @default.
- W64035408 title "Natural Polyphenols as Potent Inhibitors of DNA Methyltransferases" @default.
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