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- W66145768 endingPage "214" @default.
- W66145768 startingPage "187" @default.
- W66145768 abstract "Transdermal drug delivery has many advantages over the oral administration of drugs. This is the reason why many researchers have extensively investigated the transdermal absorption of drugs. However, a much smaller number of drugs are marketed using this route of delivery, compared to oral dosage forms, because drug absorption across the skin is very low due to the stratum corneum (the main barrier for drug absorption across the skin). Overcoming the penetration barrier would significantly improve the development of an efficient transdermal drug delivery system. Several techniques have been developed, or are under development, to bypass the stratum corneum. Approaches that have been made to overcome the stratum corneum fit into five different categories: (i) device and formulation; (ii) modification of stratum corneum by chemical enhancers; (iii) ablation; (iv) bypassing the stratum corneum via appendages; and (v) electrically assisted methods such as iontophoresis and electroporation. Furthermore, possible combinatorial uses of several approaches have been studied. Although the safety issues of these synergistic approaches still require clarification, several combinations could be promising. Finally, there is a necessity to regulate the intradermal disposition of drugs to develop a more efficient transdermal drug delivery system after overcoming the skin barrier." @default.
- W66145768 created "2016-06-24" @default.
- W66145768 creator A5053672726 @default.
- W66145768 creator A5055653919 @default.
- W66145768 creator A5085916499 @default.
- W66145768 date "2003-01-01" @default.
- W66145768 modified "2023-10-18" @default.
- W66145768 title "Strategies for Overcoming the Stratum Corneum" @default.
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