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- W71784658 abstract "Estradiol tolerates the presence of large functional groups off of the 11-beta position while retaining a reasonable relative binding affinity to Estrogen Receptor-alpha; (ER-alpha). Although RU 39,4112, a prototypical 11-beta substituted estradiol derivative, has been considered as a potent therapeutic anti-estrogen, it also has the potential for serving as a highly ER-selective targeting agent. Because there is over-expression of ER in breast cancer cells, it is a logical biological target for compounds like RU 39,411 or its analogs. In this study, I will apply this information to design and synthesize a novel and selective delivery system for breast cancer tumor cells." @default.
- W71784658 created "2016-06-24" @default.
- W71784658 creator A5077270320 @default.
- W71784658 date "2023-02-10" @default.
- W71784658 modified "2023-09-25" @default.
- W71784658 title "Rational design and synthesis of amplified therapeutic/diagnostic agents targeting the estrogen receptor" @default.
- W71784658 doi "https://doi.org/10.17760/d20401775" @default.
- W71784658 hasPublicationYear "2023" @default.
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