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- W77347164 endingPage "143" @default.
- W77347164 startingPage "130" @default.
- W77347164 abstract "Estrogen and its receptors α and β (ERα and ERβ) play a major role in tumor progression and approximately two-thirds of breast cancers express these functional receptors. Thus, the ER is a major target for current and developing therapies. Although most ER-positive tumors initially respond to hormonal therapies such as tamoxifen, many tumors will eventually become resistant to tamoxifen induced growth inhibition. This chapter will discuss molecular mechanisms that contribute to hormonal resistance of current therapies including ERα mutations, the roles of proliferation and apoptosis in tumor homeostasis and receptor coregulator proteins. Additionally, the role of nonclassical ERα signaling through growth factor receptors and the subsequent downstream-initiated signaling, and the role of the progesterone receptors will be discussed." @default.
- W77347164 created "2016-06-24" @default.
- W77347164 creator A5004815887 @default.
- W77347164 creator A5054255756 @default.
- W77347164 date "2007-01-01" @default.
- W77347164 modified "2023-10-17" @default.
- W77347164 title "Estrogen Receptors in Resistance to Hormone Therapy" @default.
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