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- W855453556 abstract "CR 2945, a receptor antagonist, was conjugated to liposome and tested for the targeting of pancreatic cancer cells in vitro. Successful conjugation was confirmed by FTIR and NMR. The size of CR 2945-conjugated liposome was about 500 nm in diameter, with the zeta-potential being -16.5 mV. In vitro anti-cancer activity of this formulation with or without gemcitabine encapsulated was tested on human pancreatic cancer cells, PANC-1. The growth inhibitory effect of gemcitabine-encapsulating CR 2945-conjugated liposome was found to be 10-fold more potent than that of gemcitabine-encapsulating non-conjugated liposome, suggesting that CR 2945 could be used as a potential cancer targeting moiety by conjugating into liposome." @default.
- W855453556 created "2016-06-24" @default.
- W855453556 date "2004-12-20" @default.
- W855453556 modified "2023-09-26" @default.
- W855453556 title "CR 2945-Conjugated Liposomes for Targeting of Human Pancreatic Cancer Cells" @default.
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- W855453556 doi "https://doi.org/10.4333/kps.2004.34.6.459" @default.
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