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- W85839286 abstract "The physicochemical properties such as solubility, partition coefficient, and membrane permeability of a drugare required for formulating and estimating drugs absorption that pass through biological membranes. Theresearch studied about solubility, partition coefficient in octanol-phosphate buffer, rabbit skin permeability andrelease from the transdermal delivery system of piroxicam with addition of 6% PVP K-30 in vitro into phosphatebuffer solution pH 7.4 at temperature 320 ± 10C. The results showed that the solubility of piroxicam was 904.44± 20.92 μg/mL. The values of log IPC and APC were 1.99 ± 0.01 and 0.08 ± 0.01, respectively. The flux,permeability coefficient, and diffusion coefficient of the piroxicam permeation process were 2.07 x 10-4μg/cm2/sec, 4.96 x 10-6 cm/minute, and 4.13 x 10-8 cm2/minute, respectively. The release mechanism ofpiroxicam from transdermal delivery system was more dominant by diffusion than erosion. The fluxes ofpiroxicam release were 0,169 and 0,107 mg/cm2/minute for formulation with 2% HPMC and 4% HPMC,respectively." @default.
- W85839286 created "2016-06-24" @default.
- W85839286 creator A5088599321 @default.
- W85839286 date "2006-08-01" @default.
- W85839286 modified "2023-09-27" @default.
- W85839286 title "The Development of Transdermal Piroxicam Using HPMC MatricesWith PVP K-30 as a Penetration Enhancer" @default.
- W85839286 hasPublicationYear "2006" @default.
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