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- W97558105 abstract "Clinical drug resistance to chemo therapeutic agents is a major obstacle for their curative potential in the treatment of human cancers. Multidrug resistance (MDR) is an important mechanism of cellular resistance to the cytotoxic activity of certain chemotherapeutic agents. Tumor cells selected for the MDR phenotype overexpress the mdr1 gene product, P-glycoprotein (P-gp), a membrane-bound drug efflux pump that confers resistance to a broad range of commonly used chemotherapeutic drugs and other agents. Numerous compounds have been identified that inhibit the efflux activity of P-gp, and reverse cellular resistance to cytotoxic agents in experimental systems [1]. This suggests that clinical drug resistance in human tumors, which often overexpress P-gp, may be potentially overcome through the concomitant administration to patients of a P-gp inhibitor with chemotherapeutic drugs." @default.
- W97558105 created "2016-06-24" @default.
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- W97558105 creator A5078696948 @default.
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- W97558105 date "1996-01-01" @default.
- W97558105 modified "2023-09-27" @default.
- W97558105 title "P-Glycoprotein-Mediated Multidrug Resistance: Experimental and Clinical Strategies for its Reversal" @default.
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