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• W984132521 abstract "ATAD2 is a bromodomain-containing protein whose overexpression is linked to poor outcomes in a number of different cancer types. To date, no potent and selective inhibitors of the bromodomain have been reported. This article describes the structure-based optimization of a series of naphthyridones from micromolar leads with no selectivity over the BET bromodomains to inhibitors with sub-100 nM ATAD2 potency and 100-fold BET selectivity." @default.
• W984132521 created "2016-06-24" @default.
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• W984132521 date "2015-07-31" @default.
• W984132521 modified "2023-10-02" @default.
• W984132521 title "Structure-Based Optimization of Naphthyridones into Potent ATAD2 Bromodomain Inhibitors" @default.
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• W984132521 doi "https://doi.org/10.1021/acs.jmedchem.5b00773" @default.
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